ARN-509 is a selective and competitive androgen receptor (AR) inhibitor (IC₅₀ = 16 nM). ARN-509 selectively binds the androgen recep tor and impairs its nuclear translocation and DNA binding to androgen response elements useful for prostate cancer tr

Numéro d'article : BIOV9535-5
Unité de mesure : 5 MG
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    ARN-509 is a selective and competitive androgen receptor (AR) inhibitor (IC₅₀ = 16 nM). ARN-509 selectively binds the androgen recep tor and impairs its nuclear translocation and DNA binding to androgen response elements useful for prostate cancer tr