GSK-269962 is a potent Rho kinase (ROCK) inhibitor (IC₅₀ values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively) . Displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases.

Item Number: BIOV9654-5
Unit of Measure: 5 MG
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    Manufacturer: BIOVISION
    Manufacturer Number: 9654-5
    Storage Temperature: Freezer (-20)

    GSK-269962 is a potent Rho kinase (ROCK) inhibitor (IC₅₀ values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively) . Displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases.